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I-Lvermectin Veterinary Medicine CAS 70288-86-7 Pharmaceutical Raw Material Powder

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I-CAS: 70288-86-7

I-1.Ivermectin iwuhlobo olusha lwe-spectrum ebanzi, esebenza kahle kakhulu, enobuthi obuphansi be-antiparasitic drug, enomphumela omuhle wokuxosha ama-parasites angaphakathi nangaphandle, ikakhulukazi ama-nematodes nama-arthropods.Kodwa-ke, ayisebenzi ngokumelene ne-cestodes, trematodes kanye ne-protozoa.Umthelela oxosha ama-macrolide antiparasitic izidakamizwa kuma-nematodes nama-arthropods usekwenyuseni ukukhululwa kwe-γ-aminobutyric acid (GABA), isidluliseli esivimbile se-Chemicalbook kanye nesibungu, kanye nokuvula iziteshi ze-Cl ion ezilawulwa yi-glutamate, okuthuthukisa ukungeneka kwemizwa. ulwelwesi oluya ku-Cl, ngaleyo ndlela luvimbele ukudluliswa kwezimpawu zemizwa futhi ekugcineni lukhubazeke izinzwa, okubangela amangqamuzana emisipha ukuba alahlekelwe amandla okufinyela, ngaleyo ndlela kuholele ekufeni kwesibungu.

I-2.Ivermectin iwuhlobo olusha lwe-semi-synthetic antibiotic insecticide, i-acaricide ne-nematicide, okuyi-ejenti ye-neurotoxic yezinambuzane kanye ne-biological penetrant.Indlela yokusebenza iwukuphazamisa imisebenzi ye-neurophysiological yezinambuzane, ikhuthaze i-Chemicalbook ukuthi ikhulule i-γ-aminobutyric acid, esebenza kumalunga ezinzwa nemisipha, ikhuphule ukukhululwa kwama-ion e-chloride, ivimbele ukudluliswa kolwazi kwamalunga ezinzwa, okuholela ekukhubazekeni. kanye nokufa okunobuthi kwezinambuzane nezibungu.

3.I-crystalline powder emhlophe noma ephuzi kancane, encibilika ku-methanol, esters nama-hydrocarbon anephunga elimnandi, engancibiliki emanzini.Igama lesiNgisi elithi Ivermectin: Ivermectin, isidakamizwa esilwa namagciwane, inomsebenzi wokuxosha ngokumelene nama-nematode, izinambuzane nezibungu.Imijovo namaphilisi enziwe nge-ivermectin asetshenziswa kakhulu ekwelapheni ama-nematode emathunjini, izimpethu ze-bull fly, izimpethu ze-striated fly, izimpethu zempumulo ekhaleni lezimvu kanye nengulube kanye nezibungu ze-Chemicalbook izimvu zomhlambi ezilwaneni ezifuywayo.Ngaphezu kwalokho, i-ivermectin ingasetshenziswa futhi ekwelapheni ama-nematodes angama-parasitic (njenge-roundworms, i-lung nematodes, njll.) ezinkukhu.Ingenziwa futhi ibe isibulala-zinambuzane sezolimo kanye ne-acaricide, esetshenziselwa ukubulala izimbuzane, amabhu amancane emifino, amabhu eklabishi, umvukuzi wamaqabunga, izintwala zokhuni, ama-nematodes, njll., amagciwane amaningi ezitshalweni.Izici ezivelele zomuthi yilezi: imiphumela emibi ekhanyayo, kanye nethamo elilodwa lomuthi kanyekanye lixosha futhi libulale izinhlobonhlobo zezimuncagazi ku-vivo kanye ne-in vitro.

Isicelo

I-1.Isebenza ngempumelelo ekwelapheni nasekulawuleni i-onchocerciasis futhi inemiphumela emibi ephansi kune-ethamazine.

2.I-Anti-parasitic, ene-anthelmintic action against nematodes, hookworms, roundworms, izikelemu, izinambuzane nezibungu.


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